C-8813
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Formula | C20H26BrNOS |
Molar mass | 408.40g·mol−1 |
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C-8813(thiobromadol) is a potentμ-opioid receptoragonistwith a distinctive chemical structure which is not closely related to other established families of opioid drugs. Thetrans-isomer was found to be around 591 times more potent thanmorphinein animal studies.[1]The same study assigned a potency of 504 times that of morphine to the related compoundBDPC.
C-8813 is claimed to be similarly potent at theδ-opioid receptor,which antagonizes the μ-induced depression of breathing, presumably making the drug safer.[1]
C-8813 has never been approved for use in humans.[citation needed]