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WKP|Q16735186
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20241121000150.0 |
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(WKP)Q16735186
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0000-0002-2397-0443
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orcid
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57034598400
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scopus
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(OCoLC)Q16735186
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US
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19000000
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Richard Lee
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American cardiac surgeon (21st century)
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1
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iso5218
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ريتشارد لي
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جراح من الولايات المتحدة الأمريكية
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Richard Lee
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siruhano Merikano
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pap
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Ричард Ли
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ru
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Richard Lee (Cardiac Surgeon)
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Amerikaans chirurg
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nl
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Richard Lee
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chirurgien américain (21e siècle)
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fr
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Richard Lee
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ciruxanu estauxunidense
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ast
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রিচার্ড লি
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bn
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Richard Lee
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amerikanischer Chirurg (21. Jahrhundert)
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de
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400
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ریچارد لی
‡9
fa
|
670
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‡a
Author's A Fluorescent Probe for Detecting Mycobacterium tuberculosis and Identifying Genes Critical for Cell Entry
|
670
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|
‡a
Author's A microbiological assessment of novel nitrofuranylamides as anti-tuberculosis agents
|
670
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|
|
‡a
Author's A newly discovered mycobacterial pathogen isolated from laboratory colonies of Xenopus species with lethal infections produces a novel form of mycolactone, the Mycobacterium ulcerans macrolide toxin
|
670
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‡a
Author's A pantothenate kinase from Staphylococcus aureus refractory to feedback regulation by coenzyme A.
|
670
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|
‡a
Author's A screen for and validation of prodrug antimicrobials
|
670
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|
|
‡a
Author's A simple in vitro PK/PD model system to determine time-kill curves of drugs against Mycobacteria
|
670
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|
|
‡a
Author's A statistical framework to evaluate virtual screening
|
670
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|
|
‡a
Author's A therapeutic approach to pantothenate kinase associated neurodegeneration
|
670
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|
|
‡a
Author's Activation of Exogenous Fatty Acids to Acyl-Acyl Carrier Protein Cannot Bypass FabI Inhibition in Neisseria
|
670
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‡a
Author's Acyl carrier protein is a cellular target for the antibacterial action of the pantothenamide class of pantothenate antimetabolites
|
670
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|
|
‡a
Author's Acyl-Phosphates Initiate Membrane Phospholipid Synthesis in Gram-Positive Pathogens
|
670
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‡a
Author's Acyl-sulfamates target the essential glycerol-phosphate acyltransferase (PlsY) in Gram-positive bacteria
|
670
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|
‡a
Author's Allosteric Regulation of Mammalian Pantothenate Kinase
|
670
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|
‡a
Author's Aminomethyl spectinomycins: a novel antibacterial chemotype for biothreat pathogens
|
670
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|
|
‡a
Author's Aminomethyl spectinomycins as therapeutics for drug-resistant respiratory tract and sexually transmitted bacterial infections
|
670
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|
|
‡a
Author's Analysis of Mycobacterium species for the presence of a macrolide toxin, mycolactone
|
670
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|
|
‡a
Author's Antibacterial and antitubercular activity of fosmidomycin, FR900098, and their lipophilic analogs
|
670
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|
|
‡a
Author's Antitubercular nitrofuran isoxazolines with improved pharmacokinetic properties
|
670
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|
|
‡a
Author's Applications of pharmacometrics in the clinical development and pharmacotherapy of anti-infectives
|
670
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|
|
‡a
Author's Biopharmaceutics, pharmacokinetics and pharmacodynamics of antituberculosis drugs
|
670
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‡a
Author's Catalysis and Sulfa Drug Resistance in Dihydropteroate Synthase
|
670
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‡a
Author's Characterization of the in vitro synthesized arabinan of mycobacterial cell walls
|
670
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‡a
Author's Chemical knockout of pantothenate kinase reveals the metabolic and genetic program responsible for hepatic coenzyme A homeostasis
|
670
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‡a
Author's Chemical modulation of the biological activity of reutericyclin: a membrane-active antibiotic from Lactobacillus reuteri
|
670
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‡a
Author's Combinatorial lead optimization of [1,2]-diamines based on ethambutol as potential antituberculosis preclinical candidates
|
670
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|
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‡a
Author's Comparative pharmacokinetics of spectinamide 1599 after subcutaneous and intrapulmonary aerosol administration in mice
|
670
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|
|
‡a
Author's Covalent modification of the Mycobacterium tuberculosis FAS-II dehydratase by Isoxyl and Thiacetazone
|
670
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|
|
‡a
Author's Crystal Structure of the 6-Hydroxymethyl-7,8-Dihydropterin Pyrophosphokinase•Dihydropteroate Synthase Bifunctional Enzyme from Francisella tularensis
|
670
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‡a
Author's Crystal structure of the anthrax drug target, Bacillus anthracis dihydrofolate reductase
|
670
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|
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‡a
Author's Design, synthesis and anti-tuberculosis activity of 1-adamantyl-3-heteroaryl ureas with improved in vitro pharmacokinetic properties
|
670
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|
|
‡a
Author's Design, synthesis, and evaluation of novel ethambutol analogues
|
670
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|
|
‡a
Author's Design, synthesis and microbiological evaluation of ampicillin-tetramic acid hybrid antibiotics
|
670
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|
|
‡a
Author's Detection of Mycolactone A/B in Mycobacterium ulcerans-Infected Human Tissue
|
670
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|
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‡a
Author's Development of a pterin-based fluorescent probe for screening dihydropteroate synthase
|
670
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‡a
Author's Development of an etoposide prodrug for dual prodrug-enzyme antitumor therapy.
|
670
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‡a
Author's Development of BODIPY FL Thalidomide As a High-Affinity Fluorescent Probe for Cereblon in a Time-Resolved Fluorescence Resonance Energy Transfer Assay
|
670
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|
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‡a
Author's Development of BODIPY FL vindoline as a novel and high-affinity pregnane X receptor fluorescent probe
|
670
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|
|
‡a
Author's Discovery and Characterization of the Antimetabolite Action of Thioacetamide-Linked 1,2,3-Triazoles as Disruptors of Cysteine Biosynthesis in Gram-Negative Bacteria
|
670
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‡a
Author's Discovery of non-carbohydrate inhibitors of aminoglycoside-modifying enzymes
|
670
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‡a
Author's Discovery of novel bacterial elongation condensing enzyme inhibitors by virtual screening
|
670
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|
|
‡a
Author's Discovery of novel isoxazolines as anti-tuberculosis agents
|
670
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|
|
‡a
Author's Discovery of novel selective inhibitors of human intestinal carboxylesterase for the amelioration of irinotecan-induced diarrhea: synthesis, quantitative structure-activity relationship analysis, and biological activity
|
670
|
|
|
‡a
Author's Discovery, synthesis, and biological evaluation of piperidinol analogs with anti-tuberculosis activity
|
670
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|
|
‡a
Author's Evaluation of analogs of reutericyclin as prospective candidates for treatment of staphylococcal skin infections
|
670
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|
|
‡a
Author's Evaluation of flavonoid and resveratrol chemical libraries reveals abyssinone II as a promising antibacterial lead
|
670
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|
|
‡a
Author's Exposure of Methicillin-Resistant Staphylococcus aureus to Low Levels of the Antibacterial THAM-3ΦG Generates a Small Colony Drug-Resistant Phenotype.
|
670
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‡a
Author's First cultivation and characterization of Mycobacterium ulcerans from the environment
|
670
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‡a
Author's Gastrointestinal localization of metronidazole by a lactobacilli-inspired tetramic acid motif improves treatment outcomes in the hamster model of Clostridium difficile infection
|
670
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|
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‡a
Author's Genome-wide expression profiling of the response to ciclopirox olamine in Candida albicans
|
670
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|
|
‡a
Author's Giant plasmid-encoded polyketide synthases produce the macrolide toxin of Mycobacterium ulcerans
|
670
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|
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‡a
Author's Globally distributed mycobacterial fish pathogens produce a novel plasmid-encoded toxic macrolide, mycolactone F
|
670
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|
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‡a
Author's Heterogeneity of mycolactones produced by clinical isolates of Mycobacterium ulcerans: implications for virulence
|
670
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|
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‡a
Author's Identification and characterization of an allosteric inhibitory site on dihydropteroate synthase
|
670
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|
|
‡a
Author's Identification of a gene involved in the biosynthesis of cyclopropanated mycolic acids in Mycobacterium tuberculosis
|
670
|
|
|
‡a
Author's In vitro and in vivo activities of HPi1, a selective antimicrobial against Helicobacter pylori
|
670
|
|
|
‡a
Author's In vitro and in vivo Evaluation of Synergism between Anti-Tubercular Spectinamides and Non-Classical Tuberculosis Antibiotics
|
670
|
|
|
‡a
Author's In vitro pharmacokinetic/pharmacodynamic models in anti-infective drug development: focus on TB
|
670
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|
|
‡a
Author's Inhibition of mycolic acid transport across the Mycobacterium tuberculosis plasma membrane
|
670
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|
|
‡a
Author's Inhibition of UDP-Gal Mutase and Mycobacterial Galactan Biosynthesis by Pyrrolidine Analogues of Galactofuranose
|
670
|
|
|
‡a
Author's Isoniazid affects multiple components of the type II fatty acid synthase system of Mycobacterium tuberculosis.
|
670
|
|
|
‡a
Author's LipE guided discovery of isopropylphenyl pyridazines as pantothenate kinase modulators
|
670
|
|
|
‡a
Author's Mechanisms involved in the intrinsic isoniazid resistance of Mycobacterium avium
|
670
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|
|
‡a
Author's Mechanisms of Resistance Associated with the Inhibition of the Dehydration Step of Type II Fatty Acid Synthase in Mycobacterium tuberculosis
|
670
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|
|
‡a
Author's Metabolic activation of CaMKII by coenzyme A.
|
670
|
|
|
‡a
Author's Methods for acquisition and assignment of multidimensional high-resolution magic angle spinning NMR of whole cell bacteria
|
670
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|
|
‡a
Author's Model-Based Exposure-Response Assessment for Spectinamide 1810 in a Mouse Model of Tuberculosis
|
670
|
|
|
‡a
Author's Mycobacterial arabinan biosynthesis: the use of synthetic arabinoside acceptors in the development of an arabinosyl transfer assay
|
670
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|
|
‡a
Author's Mycolactone: a polyketide toxin from Mycobacterium ulcerans required for virulence
|
670
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|
|
‡a
Author's Mycolic acid biosynthesis: definition and targeting of the Claisen condensation step
|
670
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|
|
‡a
Author's Mycolic acids: structure, biosynthesis and physiological functions
|
670
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|
|
‡a
Author's N-substituted 3-acetyltetramic acid derivatives as antibacterial agents
|
670
|
|
|
‡a
Author's New agents for the treatment of drug-resistant Mycobacterium tuberculosis
|
670
|
|
|
‡a
Author's Nitrofurans as novel anti-tuberculosis agents: identification, development and evaluation
|
670
|
|
|
‡a
Author's Novel acyl phosphate mimics that target PlsY, an essential acyltransferase in gram-positive bacteria
|
670
|
|
|
‡a
Author's Novel inhibitors of an emerging target in Mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesis
|
670
|
|
|
‡a
Author's Novel insights into the mechanism of inhibition of MmpL3, a target of multiple pharmacophores in Mycobacterium tuberculosis
|
670
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|
|
‡a
Author's Novel Polyoxyethylene-Containing Glycolipids Are Synthesized in Corynebacterium matruchotii and Mycobacterium smegmatis Cultured in the Presence of Tween 80.
|
670
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‡a
Author's Pantothenamides are potent, on-target inhibitors of Plasmodium falciparum growth when serum pantetheinase is inactivated
|
670
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|
|
‡a
Author's Pentacyclic nitrofurans that rapidly kill nifurtimox-resistant trypanosomes
|
670
|
|
|
‡a
Author's Pentacyclic nitrofurans with in vivo efficacy and activity against nonreplicating Mycobacterium tuberculosis
|
670
|
|
|
‡a
Author's Pharmacokinetically-guided lead optimization of nitrofuranylamide anti-tuberculosis agents
|
670
|
|
|
‡a
Author's Phase II Metabolic Pathways of Spectinamide Antitubercular Agents: A Comparative Study of the Reactivity of 4-Substituted Pyridines to Glutathione Conjugation
|
670
|
|
|
‡a
Author's Potentiation of azole antifungals by 2-adamantanamine
|
670
|
|
|
‡a
Author's Pterin-sulfa conjugates as dihydropteroate synthase inhibitors and antibacterial agents
|
670
|
|
|
‡a
Author's Quantitative structure-activity relationship studies on nitrofuranyl anti-tubercular agents
|
670
|
|
|
‡a
Author's Rapid structural characterization of the arabinogalactan and lipoarabinomannan in live mycobacterial cells using 2D and 3D HR-MAS NMR: structural changes in the arabinan due to ethambutol treatment and gene mutation are observed
|
670
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|
|
‡a
Author's RelA Mutant Enterococcus faecium with Multiantibiotic Tolerance Arising in an Immunocompromised Host
|
670
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|
|
‡a
Author's Replacing sulfa drugs with novel DHPS inhibitors
|
670
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|
|
‡a
Author's Reutericyclin and related analogues kill stationary phase Clostridium difficile at achievable colonic concentrations
|
670
|
|
|
‡a
Author's SB-224289 Antagonizes the Antifungal Mechanism of the Marine Depsipeptide Papuamide A
|
670
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|
|
‡a
Author's Screening a library of 1600 adamantyl ureas for anti-Mycobacterium tuberculosis activity in vitro and for better physical chemical properties for bioavailability
|
670
|
|
|
‡a
Author's Solid-phase synthesis and biological evaluation of a uridinyl branched peptide urea library
|
670
|
|
|
‡a
Author's Solid-phase synthesis of a thymidinyl dipeptide urea library
|
670
|
|
|
‡a
Author's Spectinamides: a new class of semisynthetic antituberculosis agents that overcome native drug efflux
|
670
|
|
|
‡a
Author's Spectinamides are effective partner agents for the treatment of tuberculosis in multiple mouse infection models
|
670
|
|
|
‡a
Author's Structural and In Vivo Studies on Trehalose-6-Phosphate Synthase from Pathogenic Fungi Provide Insights into Its Catalytic Mechanism, Biological Necessity, and Potential for Novel Antifungal Drug Design
|
670
|
|
|
‡a
Author's Structural basis for substrate recognition and chemical inhibition of oncogenic MAGE ubiquitin ligases
|
670
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|
|
‡a
Author's Structural Characterization of the Mycobacterium tuberculosis Biotin Biosynthesis Enzymes 7,8-Diaminopelargonic Acid Synthase and Dethiobiotin Synthetase,
|
670
|
|
|
‡a
Author's Structural Studies of Pterin-Based Inhibitors of Dihydropteroate Synthase
|
670
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|
|
‡a
Author's Structure-activity relationships and enzyme inhibition of pantothenamide-type pantothenate kinase inhibitors
|
670
|
|
|
‡a
Author's Structure-Activity Relationships of Spectinamide Antituberculosis Agents: A Dissection of Ribosomal Inhibition and Native Efflux Avoidance Contributions
|
670
|
|
|
‡a
Author's Structure-Based Design of Novel Pyrimido[4,5-c]pyridazine Derivatives as Dihydropteroate Synthase Inhibitors with Increased Affinity
|
670
|
|
|
‡a
Author's Structure-Based Design, Synthesis, and Evaluation of 2′-(2-Hydroxyethyl)-2′-deoxyadenosine and the 5′-Diphosphate Derivative as Ribonucleotide Reductase Inhibitors
|
670
|
|
|
‡a
Author's Syntheses and evaluation of macrocyclic engelhardione analogs as antitubercular and antibacterial agents
|
670
|
|
|
‡a
Author's Synthesis and evaluation of cyclic secondary amine substituted phenyl and benzyl nitrofuranyl amides as novel antituberculosis agents
|
670
|
|
|
‡a
Author's Synthesis and evaluation of esters and carbamates to identify critical functional groups for esterase-specific metabolism
|
670
|
|
|
‡a
Author's Synthesis and evaluation of nitrofuranylamides as novel antituberculosis agents
|
670
|
|
|
‡a
Author's Synthesis and evaluation of pretomanid (PA-824) oxazolidinone hybrids
|
670
|
|
|
‡a
Author's Synthesis and Evaluation of Thiazolidine Amide and N-Thiazolyl Amide Fluoroquinolone Derivatives.
|
670
|
|
|
‡a
Author's Synthesis and Structure–Activity Relationship of Thioacetamide-Triazoles against Escherichia coli
|
670
|
|
|
‡a
Author's Synthesis and structure of mycolactone E isolated from frog mycobacterium
|
670
|
|
|
‡a
Author's Synthesis of beta-D-arabinofuranosyl-1-monophosphoryl polyprenols: examination of their function as mycobacterial arabinosyl transferase donors.
|
670
|
|
|
‡a
Author's Synthesis of bi-substrate state mimics of dihydropteroate synthase as potential inhibitors and molecular probes
|
670
|
|
|
‡a
Author's Synthesis of new and potent analogues of anti-tuberculosis agent 5-nitro-furan-2-carboxylic acid 4-
|
670
|
|
|
‡a
Author's Synthesis of new and potent analogues of anti-tuberculosis agent 5-nitro-furan-2-carboxylic acid 4-(4-benzyl-piperazin-1-yl)-benzylamide with improved bioavailability
|
670
|
|
|
‡a
Author's Synthesis, optimization and structure-activity relationships of 3,5-disubstituted isoxazolines as new anti-tuberculosis agents
|
670
|
|
|
‡a
Author's Synthesis, structure-activity relationship studies, and antibacterial evaluation of 4-chromanones and chalcones, as well as olympicin A and derivatives
|
670
|
|
|
‡a
Author's Targeting bacterial membrane function: an underexploited mechanism for treating persistent infections
|
670
|
|
|
‡a
Author's The identification, analysis and structure-based development of novel inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase
|
670
|
|
|
‡a
Author's The membrane as a target for controlling hypervirulent Clostridium difficile infections
|
670
|
|
|
‡a
Author's The structure-activity relationship of urea derivatives as anti-tuberculosis agents
|
670
|
|
|
‡a
Author's The structure of the pantothenate kinase.ADP.pantothenate ternary complex reveals the relationship between the binding sites for substrate, allosteric regulator, and antimetabolites
|
670
|
|
|
‡a
Author's Therapeutic Potential of the Mycobacterium tuberculosis Mycolic Acid Transporter, MmpL3
|
670
|
|
|
‡a
Author's Topology and Active Site of PlsY
|
670
|
|
|
‡a
Author's Ureadepsipeptides as ClpP Activators
|
670
|
|
|
‡a
Author's Validation of molecular docking programs for virtual screening against dihydropteroate synthase
|
670
|
|
|
‡a
wikidata site links
‡u
https://en.wikipedia.org/wiki/Richard_Lee_(surgeon)
|
909
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‡a
(orcid) 0000000223970443
‡9
1
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909
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(scopus) 57034598400
‡9
1
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919
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fluorescentprobefordetectingmycobacteriumtuberculosisandidentifyinggenescriticalforcellentry
‡A
A Fluorescent Probe for Detecting Mycobacterium tuberculosis and Identifying Genes Critical for Cell Entry
‡9
1
|
919
|
|
|
‡a
microbiologicalassessmentofnovelnitrofuranylamidesasantituberculosisagents
‡A
A microbiological assessment of novel nitrofuranylamides as anti-tuberculosis agents
‡9
1
|
919
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|
|
‡a
newlydiscoveredmycobacterialpathogenisolatedfromlaboratorycoloniesofxenopusspecieswithlethalinfectionsproducesanovelformofmycolactonethemycobacteriumulceransmacrolidetoxin
‡A
A newly discovered mycobacterial pathogen isolated from laboratory colonies of Xenopus species with lethal infections produces a novel form of mycolactone, the Mycobacterium ulcerans macrolide toxin
‡9
1
|
919
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‡a
pantothenatekinasefromstaphylococcusaureusrefractorytofeedbackregulationbycoenzymea
‡A
A pantothenate kinase from Staphylococcus aureus refractory to feedback regulation by coenzyme A.
‡9
1
|
919
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‡a
screenforandvalidationofprodrugantimicrobials
‡A
A screen for and validation of prodrug antimicrobials
‡9
1
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919
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‡a
simpleinvitropkpdmodelsystemtodeterminetimekillcurvesofdrugsagainstmycobacteria
‡A
A simple in vitro PK/PD model system to determine time-kill curves of drugs against Mycobacteria
‡9
1
|
919
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|
‡a
statisticalframeworktoevaluatevirtualscreening
‡A
A statistical framework to evaluate virtual screening
‡9
1
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919
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‡a
therapeuticapproachtopantothenatekinaseassociatedneurodegeneration
‡A
A therapeutic approach to pantothenate kinase associated neurodegeneration
‡9
1
|
919
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|
‡a
activationofexogenousfattyacidstoacylacylcarrierproteincannotbypassfabiinhibitioninneisseria
‡A
Activation of Exogenous Fatty Acids to Acyl-Acyl Carrier Protein Cannot Bypass FabI Inhibition in Neisseria
‡9
1
|
919
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‡a
acylcarrierproteinisacellulartargetfortheantibacterialactionofthepantothenamideclassofpantothenateantimetabolites
‡A
Acyl carrier protein is a cellular target for the antibacterial action of the pantothenamide class of pantothenate antimetabolites
‡9
1
|
919
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‡a
acylphosphatesinitiatemembranephospholipidsynthesisingrampositivepathogens
‡A
Acyl-Phosphates Initiate Membrane Phospholipid Synthesis in Gram-Positive Pathogens
‡9
1
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919
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‡a
acylsulfamatestargettheessentialglycerolphosphateacyltransferaseplsyingrampositivebacteria
‡A
Acyl-sulfamates target the essential glycerol-phosphate acyltransferase (PlsY) in Gram-positive bacteria
‡9
1
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919
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‡a
allostericregulationofmammalianpantothenatekinase
‡A
Allosteric Regulation of Mammalian Pantothenate Kinase
‡9
1
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919
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‡a
aminomethylspectinomycinsanovelantibacterialchemotypeforbiothreatpathogens
‡A
Aminomethyl spectinomycins: a novel antibacterial chemotype for biothreat pathogens
‡9
1
|
919
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‡a
aminomethylspectinomycinsastherapeuticsfordrugresistantrespiratorytractandsexuallytransmittedbacterialinfections
‡A
Aminomethyl spectinomycins as therapeutics for drug-resistant respiratory tract and sexually transmitted bacterial infections
‡9
1
|
919
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‡a
analysisofmycobacteriumspeciesforthepresenceofamacrolidetoxinmycolactone
‡A
Analysis of Mycobacterium species for the presence of a macrolide toxin, mycolactone
‡9
1
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919
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‡a
antibacterialandantitubercularactivityoffosmidomycinfr900098andtheirlipophilicanalogs
‡A
Antibacterial and antitubercular activity of fosmidomycin, FR900098, and their lipophilic analogs
‡9
1
|
919
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‡a
antitubercularnitrofuranisoxazolineswithimprovedpharmacokineticproperties
‡A
Antitubercular nitrofuran isoxazolines with improved pharmacokinetic properties
‡9
1
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919
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‡a
applicationsofpharmacometricsintheclinicaldevelopmentandpharmacotherapyofantiinfectives
‡A
Applications of pharmacometrics in the clinical development and pharmacotherapy of anti-infectives
‡9
1
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919
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‡a
biopharmaceuticspharmacokineticsandpharmacodynamicsofantituberculosisdrugs
‡A
Biopharmaceutics, pharmacokinetics and pharmacodynamics of antituberculosis drugs
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919
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|
‡a
catalysisandsulfadrugresistanceindihydropteroatesynthase
‡A
Catalysis and Sulfa Drug Resistance in Dihydropteroate Synthase
‡9
1
|
919
|
|
|
‡a
characterizationoftheinvitrosynthesizedarabinanofmycobacterialcellwalls
‡A
Characterization of the in vitro synthesized arabinan of mycobacterial cell walls
‡9
1
|
919
|
|
|
‡a
chemicalknockoutofpantothenatekinaserevealsthemetabolicandgeneticprogramresponsibleforhepaticcoenzymeahomeostasis
‡A
Chemical knockout of pantothenate kinase reveals the metabolic and genetic program responsible for hepatic coenzyme A homeostasis
‡9
1
|
919
|
|
|
‡a
chemicalmodulationofthebiologicalactivityofreutericyclinamembraneactiveantibioticfromlactobacillusreuteri
‡A
Chemical modulation of the biological activity of reutericyclin: a membrane-active antibiotic from Lactobacillus reuteri
‡9
1
|
919
|
|
|
‡a
combinatorialleadoptimizationofdiaminesbasedonethambutolaspotentialantituberculosispreclinicalcandidates
‡A
Combinatorial lead optimization of [1,2]-diamines based on ethambutol as potential antituberculosis preclinical candidates
‡9
1
|
919
|
|
|
‡a
comparativepharmacokineticsofspectinamide1599aftersubcutaneousandintrapulmonaryaerosoladministrationinmice
‡A
Comparative pharmacokinetics of spectinamide 1599 after subcutaneous and intrapulmonary aerosol administration in mice
‡9
1
|
919
|
|
|
‡a
covalentmodificationofthemycobacteriumtuberculosisfas2dehydratasebyisoxylandthiacetazone
‡A
Covalent modification of the Mycobacterium tuberculosis FAS-II dehydratase by Isoxyl and Thiacetazone
‡9
1
|
919
|
|
|
‡a
crystalstructureofthe6hydroxymethyl78dihydropterinpyrophosphokinasedihydropteroatesynthasebifunctionalenzymefromfrancisellatularensis
‡A
Crystal Structure of the 6-Hydroxymethyl-7,8-Dihydropterin Pyrophosphokinase•Dihydropteroate Synthase Bifunctional Enzyme from Francisella tularensis
‡9
1
|
919
|
|
|
‡a
crystalstructureoftheanthraxdrugtargetbacillusanthracisdihydrofolatereductase
‡A
Crystal structure of the anthrax drug target, Bacillus anthracis dihydrofolate reductase
‡9
1
|
919
|
|
|
‡a
designsynthesisandantituberculosisactivityof1adamantyl3heteroarylureaswithimprovedinvitropharmacokineticproperties
‡A
Design, synthesis and anti-tuberculosis activity of 1-adamantyl-3-heteroaryl ureas with improved in vitro pharmacokinetic properties
‡9
1
|
919
|
|
|
‡a
designsynthesisandevaluationofnovelethambutolanalogues
‡A
Design, synthesis, and evaluation of novel ethambutol analogues
‡9
1
|
919
|
|
|
‡a
designsynthesisandmicrobiologicalevaluationofampicillintetramicacidhybridantibiotics
‡A
Design, synthesis and microbiological evaluation of ampicillin-tetramic acid hybrid antibiotics
‡9
1
|
919
|
|
|
‡a
detectionofmycolactoneabinmycobacteriumulceransinfectedhumantissue
‡A
Detection of Mycolactone A/B in Mycobacterium ulcerans-Infected Human Tissue
‡9
1
|
919
|
|
|
‡a
developmentofapterinbasedfluorescentprobeforscreeningdihydropteroatesynthase
‡A
Development of a pterin-based fluorescent probe for screening dihydropteroate synthase
‡9
1
|
919
|
|
|
‡a
developmentofanetoposideprodrugfordualprodrugenzymeantitumortherapy
‡A
Development of an etoposide prodrug for dual prodrug-enzyme antitumor therapy.
‡9
1
|
919
|
|
|
‡a
developmentofbodipyflthalidomideasahighaffinityfluorescentprobeforcerebloninatimeresolvedfluorescenceresonanceenergytransferassay
‡A
Development of BODIPY FL Thalidomide As a High-Affinity Fluorescent Probe for Cereblon in a Time-Resolved Fluorescence Resonance Energy Transfer Assay
‡9
1
|
919
|
|
|
‡a
developmentofbodipyflvindolineasanovelandhighaffinitypregnane10receptorfluorescentprobe
‡A
Development of BODIPY FL vindoline as a novel and high-affinity pregnane X receptor fluorescent probe
‡9
1
|
919
|
|
|
‡a
discoveryandcharacterizationoftheantimetaboliteactionofthioacetamidelinked123triazolesasdisruptorsofcysteinebiosynthesisingramnegativebacteria
‡A
Discovery and Characterization of the Antimetabolite Action of Thioacetamide-Linked 1,2,3-Triazoles as Disruptors of Cysteine Biosynthesis in Gram-Negative Bacteria
‡9
1
|
919
|
|
|
‡a
discoveryofnoncarbohydrateinhibitorsofaminoglycosidemodifyingenzymes
‡A
Discovery of non-carbohydrate inhibitors of aminoglycoside-modifying enzymes
‡9
1
|
919
|
|
|
‡a
discoveryofnovelbacterialelongationcondensingenzymeinhibitorsbyvirtualscreening
‡A
Discovery of novel bacterial elongation condensing enzyme inhibitors by virtual screening
‡9
1
|
919
|
|
|
‡a
discoveryofnovelisoxazolinesasantituberculosisagents
‡A
Discovery of novel isoxazolines as anti-tuberculosis agents
‡9
1
|
919
|
|
|
‡a
discoveryofnovelselectiveinhibitorsofhumanintestinalcarboxylesterasefortheameliorationofirinotecaninduceddiarrheasynthesisquantitativestructureactivityrelationshipanalysisandbiologicalactivity
‡A
Discovery of novel selective inhibitors of human intestinal carboxylesterase for the amelioration of irinotecan-induced diarrhea: synthesis, quantitative structure-activity relationship analysis, and biological activity
‡9
1
|
919
|
|
|
‡a
discoverysynthesisandbiologicalevaluationofpiperidinolanalogswithantituberculosisactivity
‡A
Discovery, synthesis, and biological evaluation of piperidinol analogs with anti-tuberculosis activity
‡9
1
|
919
|
|
|
‡a
evaluationofanalogsofreutericyclinasprospectivecandidatesfortreatmentofstaphylococcalskininfections
‡A
Evaluation of analogs of reutericyclin as prospective candidates for treatment of staphylococcal skin infections
‡9
1
|
919
|
|
|
‡a
evaluationofflavonoidandresveratrolchemicallibrariesrevealsabyssinone2asapromisingantibacteriallead
‡A
Evaluation of flavonoid and resveratrol chemical libraries reveals abyssinone II as a promising antibacterial lead
‡9
1
|
919
|
|
|
‡a
exposureofmethicillinresistantstaphylococcusaureustolowlevelsoftheantibacterialtham3φggeneratesasmallcolonydrugresistantphenotype
‡A
Exposure of Methicillin-Resistant Staphylococcus aureus to Low Levels of the Antibacterial THAM-3ΦG Generates a Small Colony Drug-Resistant Phenotype.
‡9
1
|
919
|
|
|
‡a
1cultivationandcharacterizationofmycobacteriumulceransfromtheenvironment
‡A
First cultivation and characterization of Mycobacterium ulcerans from the environment
‡9
1
|
919
|
|
|
‡a
gastrointestinallocalizationofmetronidazolebyalactobacilliinspiredtetramicacidmotifimprovestreatmentoutcomesinthehamstermodelofclostridiumdifficileinfection
‡A
Gastrointestinal localization of metronidazole by a lactobacilli-inspired tetramic acid motif improves treatment outcomes in the hamster model of Clostridium difficile infection
‡9
1
|
919
|
|
|
‡a
genomewideexpressionprofilingoftheresponsetociclopiroxolamineincandidaalbicans
‡A
Genome-wide expression profiling of the response to ciclopirox olamine in Candida albicans
‡9
1
|
919
|
|
|
‡a
giantplasmidencodedpolyketidesynthasesproducethemacrolidetoxinofmycobacteriumulcerans
‡A
Giant plasmid-encoded polyketide synthases produce the macrolide toxin of Mycobacterium ulcerans
‡9
1
|
919
|
|
|
‡a
globallydistributedmycobacterialfishpathogensproduceanovelplasmidencodedtoxicmacrolidemycolactonef
‡A
Globally distributed mycobacterial fish pathogens produce a novel plasmid-encoded toxic macrolide, mycolactone F
‡9
1
|
919
|
|
|
‡a
heterogeneityofmycolactonesproducedbyclinicalisolatesofmycobacteriumulceransimplicationsforvirulence
‡A
Heterogeneity of mycolactones produced by clinical isolates of Mycobacterium ulcerans: implications for virulence
‡9
1
|
919
|
|
|
‡a
identificationandcharacterizationofanallostericinhibitorysiteondihydropteroatesynthase
‡A
Identification and characterization of an allosteric inhibitory site on dihydropteroate synthase
‡9
1
|
919
|
|
|
‡a
identificationofageneinvolvedinthebiosynthesisofcyclopropanatedmycolicacidsinmycobacteriumtuberculosis
‡A
Identification of a gene involved in the biosynthesis of cyclopropanated mycolic acids in Mycobacterium tuberculosis
‡9
1
|
919
|
|
|
‡a
invitroandinvivoactivitiesofhpi1aselectiveantimicrobialagainsthelicobacterpylori
‡A
In vitro and in vivo activities of HPi1, a selective antimicrobial against Helicobacter pylori
‡9
1
|
919
|
|
|
‡a
invitroandinvivoevaluationofsynergismbetweenantitubercularspectinamidesandnonclassicaltuberculosisantibiotics
‡A
In vitro and in vivo Evaluation of Synergism between Anti-Tubercular Spectinamides and Non-Classical Tuberculosis Antibiotics
‡9
1
|
919
|
|
|
‡a
invitropharmacokineticpharmacodynamicmodelsinantiinfectivedrugdevelopmentfocusontb
‡A
In vitro pharmacokinetic/pharmacodynamic models in anti-infective drug development: focus on TB
‡9
1
|
919
|
|
|
‡a
inhibitionofmycolicacidtransportacrossthemycobacteriumtuberculosisplasmamembrane
‡A
Inhibition of mycolic acid transport across the Mycobacterium tuberculosis plasma membrane
‡9
1
|
919
|
|
|
‡a
inhibitionofudpgalmutaseandmycobacterialgalactanbiosynthesisbypyrrolidineanaloguesofgalactofuranose
‡A
Inhibition of UDP-Gal Mutase and Mycobacterial Galactan Biosynthesis by Pyrrolidine Analogues of Galactofuranose
‡9
1
|
919
|
|
|
‡a
isoniazidaffectsmultiplecomponentsofthetype2fattyacidsynthasesystemofmycobacteriumtuberculosis
‡A
Isoniazid affects multiple components of the type II fatty acid synthase system of Mycobacterium tuberculosis.
‡9
1
|
919
|
|
|
‡a
lipeguideddiscoveryofisopropylphenylpyridazinesaspantothenatekinasemodulators
‡A
LipE guided discovery of isopropylphenyl pyridazines as pantothenate kinase modulators
‡9
1
|
919
|
|
|
‡a
mechanismsinvolvedintheintrinsicisoniazidresistanceofmycobacteriumavium
‡A
Mechanisms involved in the intrinsic isoniazid resistance of Mycobacterium avium
‡9
1
|
919
|
|
|
‡a
mechanismsofresistanceassociatedwiththeinhibitionofthedehydrationstepoftype2fattyacidsynthaseinmycobacteriumtuberculosis
‡A
Mechanisms of Resistance Associated with the Inhibition of the Dehydration Step of Type II Fatty Acid Synthase in Mycobacterium tuberculosis
‡9
1
|
919
|
|
|
‡a
metabolicactivationofcamkiibycoenzymea
‡A
Metabolic activation of CaMKII by coenzyme A.
‡9
1
|
919
|
|
|
‡a
methodsforacquisitionandassignmentofmultidimensionalhighresolutionmagicanglespinningnmrofwholecellbacteria
‡A
Methods for acquisition and assignment of multidimensional high-resolution magic angle spinning NMR of whole cell bacteria
‡9
1
|
919
|
|
|
‡a
modelbasedexposureresponseassessmentforspectinamide1810inamousemodeloftuberculosis
‡A
Model-Based Exposure-Response Assessment for Spectinamide 1810 in a Mouse Model of Tuberculosis
‡9
1
|
919
|
|
|
‡a
mycobacterialarabinanbiosynthesistheuseofsyntheticarabinosideacceptorsinthedevelopmentofanarabinosyltransferassay
‡A
Mycobacterial arabinan biosynthesis: the use of synthetic arabinoside acceptors in the development of an arabinosyl transfer assay
‡9
1
|
919
|
|
|
‡a
mycolactoneapolyketidetoxinfrommycobacteriumulceransrequiredforvirulence
‡A
Mycolactone: a polyketide toxin from Mycobacterium ulcerans required for virulence
‡9
1
|
919
|
|
|
‡a
mycolicacidbiosynthesisdefinitionandtargetingoftheclaisencondensationstep
‡A
Mycolic acid biosynthesis: definition and targeting of the Claisen condensation step
‡9
1
|
919
|
|
|
‡a
mycolicacidsstructurebiosynthesisandphysiologicalfunctions
‡A
Mycolic acids: structure, biosynthesis and physiological functions
‡9
1
|
919
|
|
|
‡a
nsubstituted3acetyltetramicacidderivativesasantibacterialagents
‡A
N-substituted 3-acetyltetramic acid derivatives as antibacterial agents
‡9
1
|
919
|
|
|
‡a
newagentsforthetreatmentofdrugresistantmycobacteriumtuberculosis
‡A
New agents for the treatment of drug-resistant Mycobacterium tuberculosis
‡9
1
|
919
|
|
|
‡a
nitrofuransasnovelantituberculosisagentsidentificationdevelopmentandevaluation
‡A
Nitrofurans as novel anti-tuberculosis agents: identification, development and evaluation
‡9
1
|
919
|
|
|
‡a
novelacylphosphatemimicsthattargetplsyanessentialacyltransferaseingrampositivebacteria
‡A
Novel acyl phosphate mimics that target PlsY, an essential acyltransferase in gram-positive bacteria
‡9
1
|
919
|
|
|
‡a
novelinhibitorsofanemergingtargetinmycobacteriumtuberculosissubstitutedthiazolidinonesasinhibitorsofdtdprhamnosesynthesis
‡A
Novel inhibitors of an emerging target in Mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesis
‡9
1
|
919
|
|
|
‡a
novelinsightsintothemechanismofinhibitionofmmpl3atargetofmultiplepharmacophoresinmycobacteriumtuberculosis
‡A
Novel insights into the mechanism of inhibition of MmpL3, a target of multiple pharmacophores in Mycobacterium tuberculosis
‡9
1
|
919
|
|
|
‡a
novelpolyoxyethylenecontainingglycolipidsaresynthesizedincorynebacteriummatruchotiiandmycobacteriumsmegmatisculturedinthepresenceoftween80
‡A
Novel Polyoxyethylene-Containing Glycolipids Are Synthesized in Corynebacterium matruchotii and Mycobacterium smegmatis Cultured in the Presence of Tween 80.
‡9
1
|
919
|
|
|
‡a
pantothenamidesarepotentontargetinhibitorsofplasmodiumfalciparumgrowthwhenserumpantetheinaseisinactivated
‡A
Pantothenamides are potent, on-target inhibitors of Plasmodium falciparum growth when serum pantetheinase is inactivated
‡9
1
|
919
|
|
|
‡a
pentacyclicnitrofuransthatrapidlykillnifurtimoxresistanttrypanosomes
‡A
Pentacyclic nitrofurans that rapidly kill nifurtimox-resistant trypanosomes
‡9
1
|
919
|
|
|
‡a
pentacyclicnitrofuranswithinvivoefficacyandactivityagainstnonreplicatingmycobacteriumtuberculosis
‡A
Pentacyclic nitrofurans with in vivo efficacy and activity against nonreplicating Mycobacterium tuberculosis
‡9
1
|
919
|
|
|
‡a
pharmacokineticallyguidedleadoptimizationofnitrofuranylamideantituberculosisagents
‡A
Pharmacokinetically-guided lead optimization of nitrofuranylamide anti-tuberculosis agents
‡9
1
|
919
|
|
|
‡a
phase2metabolicpathwaysofspectinamideantitubercularagentsacomparativestudyofthereactivityof4substitutedpyridinestoglutathioneconjugation
‡A
Phase II Metabolic Pathways of Spectinamide Antitubercular Agents: A Comparative Study of the Reactivity of 4-Substituted Pyridines to Glutathione Conjugation
‡9
1
|
919
|
|
|
‡a
potentiationofazoleantifungalsby2adamantanamine
‡A
Potentiation of azole antifungals by 2-adamantanamine
‡9
1
|
919
|
|
|
‡a
pterinsulfaconjugatesasdihydropteroatesynthaseinhibitorsandantibacterialagents
‡A
Pterin-sulfa conjugates as dihydropteroate synthase inhibitors and antibacterial agents
‡9
1
|
919
|
|
|
‡a
quantitativestructureactivityrelationshipstudiesonnitrofuranylantitubercularagents
‡A
Quantitative structure-activity relationship studies on nitrofuranyl anti-tubercular agents
‡9
1
|
919
|
|
|
‡a
rapidstructuralcharacterizationofthearabinogalactanandlipoarabinomannaninlivemycobacterialcellsusing2dand3dhrmasnmrstructuralchangesinthearabinanduetoethambutoltreatmentandgenemutationareobserved
‡A
Rapid structural characterization of the arabinogalactan and lipoarabinomannan in live mycobacterial cells using 2D and 3D HR-MAS NMR: structural changes in the arabinan due to ethambutol treatment and gene mutation are observed
‡9
1
|
919
|
|
|
‡a
relamutantenterococcusfaeciumwithmultiantibiotictolerancearisinginanimmunocompromisedhost
‡A
RelA Mutant Enterococcus faecium with Multiantibiotic Tolerance Arising in an Immunocompromised Host
‡9
1
|
919
|
|
|
‡a
replacingsulfadrugswithnoveldhpsinhibitors
‡A
Replacing sulfa drugs with novel DHPS inhibitors
‡9
1
|
919
|
|
|
‡a
reutericyclinandrelatedanalogueskillstationaryphaseclostridiumdifficileatachievablecolonicconcentrations
‡A
Reutericyclin and related analogues kill stationary phase Clostridium difficile at achievable colonic concentrations
‡9
1
|
919
|
|
|
‡a
sb224289antagonizestheantifungalmechanismofthemarinedepsipeptidepapuamidea
‡A
SB-224289 Antagonizes the Antifungal Mechanism of the Marine Depsipeptide Papuamide A
‡9
1
|
919
|
|
|
‡a
screeningalibraryof1600adamantylureasforantimycobacteriumtuberculosisactivityinvitroandforbetterphysicalchemicalpropertiesforbioavailability
‡A
Screening a library of 1600 adamantyl ureas for anti-Mycobacterium tuberculosis activity in vitro and for better physical chemical properties for bioavailability
‡9
1
|
919
|
|
|
‡a
solidphasesynthesisandbiologicalevaluationofauridinylbranchedpeptideurealibrary
‡A
Solid-phase synthesis and biological evaluation of a uridinyl branched peptide urea library
‡9
1
|
919
|
|
|
‡a
solidphasesynthesisofathymidinyldipeptideurealibrary
‡A
Solid-phase synthesis of a thymidinyl dipeptide urea library
‡9
1
|
919
|
|
|
‡a
spectinamidesanewclassofsemisyntheticantituberculosisagentsthatovercomenativedrugefflux
‡A
Spectinamides: a new class of semisynthetic antituberculosis agents that overcome native drug efflux
‡9
1
|
919
|
|
|
‡a
spectinamidesareeffectivepartneragentsforthetreatmentoftuberculosisinmultiplemouseinfectionmodels
‡A
Spectinamides are effective partner agents for the treatment of tuberculosis in multiple mouse infection models
‡9
1
|
919
|
|
|
‡a
structuralandinvivostudiesontrehalose6phosphatesynthasefrompathogenicfungiprovideinsightsintoitscatalyticmechanismbiologicalnecessityandpotentialfornovelantifungaldrugdesign
‡A
Structural and In Vivo Studies on Trehalose-6-Phosphate Synthase from Pathogenic Fungi Provide Insights into Its Catalytic Mechanism, Biological Necessity, and Potential for Novel Antifungal Drug Design
‡9
1
|
919
|
|
|
‡a
structuralbasisforsubstraterecognitionandchemicalinhibitionofoncogenicmageubiquitinligases
‡A
Structural basis for substrate recognition and chemical inhibition of oncogenic MAGE ubiquitin ligases
‡9
1
|
919
|
|
|
‡a
structuralcharacterizationofthemycobacteriumtuberculosisbiotinbiosynthesisenzymes78diaminopelargonicacidsynthaseanddethiobiotinsynthetase
‡A
Structural Characterization of the Mycobacterium tuberculosis Biotin Biosynthesis Enzymes 7,8-Diaminopelargonic Acid Synthase and Dethiobiotin Synthetase,
‡9
1
|
919
|
|
|
‡a
structuralstudiesofpterinbasedinhibitorsofdihydropteroatesynthase
‡A
Structural Studies of Pterin-Based Inhibitors of Dihydropteroate Synthase
‡9
1
|
919
|
|
|
‡a
structureactivityrelationshipsandenzymeinhibitionofpantothenamidetypepantothenatekinaseinhibitors
‡A
Structure-activity relationships and enzyme inhibition of pantothenamide-type pantothenate kinase inhibitors
‡9
1
|
919
|
|
|
‡a
structureactivityrelationshipsofspectinamideantituberculosisagentsadissectionofribosomalinhibitionandnativeeffluxavoidancecontributions
‡A
Structure-Activity Relationships of Spectinamide Antituberculosis Agents: A Dissection of Ribosomal Inhibition and Native Efflux Avoidance Contributions
‡9
1
|
919
|
|
|
‡a
structurebaseddesignofnovelpyrimidopyridazinederivativesasdihydropteroatesynthaseinhibitorswithincreasedaffinity
‡A
Structure-Based Design of Novel Pyrimido[4,5-c]pyridazine Derivatives as Dihydropteroate Synthase Inhibitors with Increased Affinity
‡9
1
|
919
|
|
|
‡a
structurebaseddesignsynthesisandevaluationof22hydroxyethyl2deoxyadenosineandthe5diphosphatederivativeasribonucleotidereductaseinhibitors
‡A
Structure-Based Design, Synthesis, and Evaluation of 2′-(2-Hydroxyethyl)-2′-deoxyadenosine and the 5′-Diphosphate Derivative as Ribonucleotide Reductase Inhibitors
‡9
1
|
919
|
|
|
‡a
synthesesandevaluationofmacrocyclicengelhardioneanalogsasantitubercularandantibacterialagents
‡A
Syntheses and evaluation of macrocyclic engelhardione analogs as antitubercular and antibacterial agents
‡9
1
|
919
|
|
|
‡a
synthesisandevaluationofcyclicsecondaryaminesubstitutedphenylandbenzylnitrofuranylamidesasnovelantituberculosisagents
‡A
Synthesis and evaluation of cyclic secondary amine substituted phenyl and benzyl nitrofuranyl amides as novel antituberculosis agents
‡9
1
|
919
|
|
|
‡a
synthesisandevaluationofestersandcarbamatestoidentifycriticalfunctionalgroupsforesterasespecificmetabolism
‡A
Synthesis and evaluation of esters and carbamates to identify critical functional groups for esterase-specific metabolism
‡9
1
|
919
|
|
|
‡a
synthesisandevaluationofnitrofuranylamidesasnovelantituberculosisagents
‡A
Synthesis and evaluation of nitrofuranylamides as novel antituberculosis agents
‡9
1
|
919
|
|
|
‡a
synthesisandevaluationofpretomanidpa824oxazolidinonehybrids
‡A
Synthesis and evaluation of pretomanid (PA-824) oxazolidinone hybrids
‡9
1
|
919
|
|
|
‡a
synthesisandevaluationofthiazolidineamideandnthiazolylamidefluoroquinolonederivatives
‡A
Synthesis and Evaluation of Thiazolidine Amide and N-Thiazolyl Amide Fluoroquinolone Derivatives.
‡9
1
|
919
|
|
|
‡a
synthesisandstructureactivityrelationshipofthioacetamidetriazolesagainstescherichiacoli
‡A
Synthesis and Structure–Activity Relationship of Thioacetamide-Triazoles against Escherichia coli
‡9
1
|
919
|
|
|
‡a
synthesisandstructureofmycolactoneeisolatedfromfrogmycobacterium
‡A
Synthesis and structure of mycolactone E isolated from frog mycobacterium
‡9
1
|
919
|
|
|
‡a
synthesisofbeta500arabinofuranosyl1monophosphorylpolyprenolsexaminationoftheirfunctionasmycobacterialarabinosyltransferasedonors
‡A
Synthesis of beta-D-arabinofuranosyl-1-monophosphoryl polyprenols: examination of their function as mycobacterial arabinosyl transferase donors.
‡9
1
|
919
|
|
|
‡a
synthesisofbisubstratestatemimicsofdihydropteroatesynthaseaspotentialinhibitorsandmolecularprobes
‡A
Synthesis of bi-substrate state mimics of dihydropteroate synthase as potential inhibitors and molecular probes
‡9
1
|
919
|
|
|
‡a
synthesisofnewandpotentanaloguesofantituberculosisagent5nitrofuran2carboxylicacid4
‡A
Synthesis of new and potent analogues of anti-tuberculosis agent 5-nitro-furan-2-carboxylic acid 4-
‡9
1
|
919
|
|
|
‡a
synthesisofnewandpotentanaloguesofantituberculosisagent5nitrofuran2carboxylicacid44benzylpiperazin1ylbenzylamidewithimprovedbioavailability
‡A
Synthesis of new and potent analogues of anti-tuberculosis agent 5-nitro-furan-2-carboxylic acid 4-(4-benzyl-piperazin-1-yl)-benzylamide with improved bioavailability
‡9
1
|
919
|
|
|
‡a
synthesisoptimizationandstructureactivityrelationshipsof35disubstitutedisoxazolinesasnewantituberculosisagents
‡A
Synthesis, optimization and structure-activity relationships of 3,5-disubstituted isoxazolines as new anti-tuberculosis agents
‡9
1
|
919
|
|
|
‡a
synthesisstructureactivityrelationshipstudiesandantibacterialevaluationof4chromanonesandchalconesaswellasolympicinaandderivatives
‡A
Synthesis, structure-activity relationship studies, and antibacterial evaluation of 4-chromanones and chalcones, as well as olympicin A and derivatives
‡9
1
|
919
|
|
|
‡a
targetingbacterialmembranefunctionanunderexploitedmechanismfortreatingpersistentinfections
‡A
Targeting bacterial membrane function: an underexploited mechanism for treating persistent infections
‡9
1
|
919
|
|
|
‡a
identificationanalysisandstructurebaseddevelopmentofnovelinhibitorsof6hydroxymethyl78dihydropterinpyrophosphokinase
‡A
The identification, analysis and structure-based development of novel inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase
‡9
1
|
919
|
|
|
‡a
membraneasatargetforcontrollinghypervirulentclostridiumdifficileinfections
‡A
The membrane as a target for controlling hypervirulent Clostridium difficile infections
‡9
1
|
919
|
|
|
‡a
structureactivityrelationshipofureaderivativesasantituberculosisagents
‡A
The structure-activity relationship of urea derivatives as anti-tuberculosis agents
‡9
1
|
919
|
|
|
‡a
structureofthepantothenatekinaseadppantothenateternarycomplexrevealstherelationshipbetweenthebindingsitesforsubstrateallostericregulatorandantimetabolites
‡A
The structure of the pantothenate kinase.ADP.pantothenate ternary complex reveals the relationship between the binding sites for substrate, allosteric regulator, and antimetabolites
‡9
1
|
919
|
|
|
‡a
therapeuticpotentialofthemycobacteriumtuberculosismycolicacidtransportermmpl3
‡A
Therapeutic Potential of the Mycobacterium tuberculosis Mycolic Acid Transporter, MmpL3
‡9
1
|
919
|
|
|
‡a
topologyandactivesiteofplsy
‡A
Topology and Active Site of PlsY
‡9
1
|
919
|
|
|
‡a
ureadepsipeptidesasclppactivators
‡A
Ureadepsipeptides as ClpP Activators
‡9
1
|
919
|
|
|
‡a
validationofmoleculardockingprogramsforvirtualscreeningagainstdihydropteroatesynthase
‡A
Validation of molecular docking programs for virtual screening against dihydropteroate synthase
‡9
1
|
946
|
|
|
‡a
b
‡9
1
|
947
|
|
|
‡a
US
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1
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996
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LC|n 85042235
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LIH|LNB:B_g__o__d_;=CG
|
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ISNI|0000000000830013
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CAOONL|ncf11324323
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LC|no2011061474
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ISNI|0000000022371962
|
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|
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NUKAT|n 2011108202
|
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LC|no2010197687
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CAOONL|ncf11335371
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CAOONL|ncf10257099
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ISNI|0000000115428307
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CAOONL|ncf11370248
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LC|no 00043263
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LC|n 2004011731
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LC|n 88185489
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J9U|987007460307005171
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J9U|987007389035705171
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NII|DA10894801
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BNF|12347122
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LC|n 84150447
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DNB|173356214
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ISNI|0000000108686527
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LC|n 00097833
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LC|n 88111956
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NTA|306972778
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LC|n 2022065844
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SUDOC|070347328
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ISNI|0000000042107448
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LNB|LNC10-000012365
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ISNI|0000000491696145
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J9U|987012329603605171
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LC|no2011062458
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LC|no2010176341
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LIH|LNB:BDJ6;=_q_P
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SUDOC|172520983
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DNB|1067795618
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LC|n 90622043
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NTA|174340818
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LC|no2014036171
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LC|n 88619456
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JPG|500280978
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NII|DA02305315
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NLR|RU NLR AUTH 771263
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SUDOC|171553020
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ISNI|0000000076283087
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ISNI|0000000055378722
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BNF|12479623
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ISNI|0000000136073322
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NII|DA06775161
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NII|DA13257713
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CAOONL|ncf10970719
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RERO|A000103615
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LC|n 85020519
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NKC|jcu2014802131
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BIBSYS|90528112
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J9U|987007379315105171
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ISNI|0000000460541511
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LC|n 84111796
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RERO|A017533835
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BIBSYS|2003193
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JPG|500111609
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LC|n 82125985
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LC|n 78090953
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ISNI|0000000075565728
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JPG|500253245
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NTA|141934972
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SUDOC|149474113
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996
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LC|n 82093298
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DNB|1155025172
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BIBSYS|90375609
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SUDOC|200616013
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BIBSYS|90589616
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NTA|381355888
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J9U|987007316230505171
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NUKAT|n 2006118869
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DNB|119451050
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LC|n 84212495
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BIBSYS|90271538
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NTA|148448674
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996
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DNB|122853393
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LC|n 81127867
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LC|n 84087754
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LC|n 86031023
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ISNI|0000000039407677
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ISNI|0000000497037917
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NLR|RU NLR AUTH 771262
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996
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BIBSYS|90342269
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LC|n 79091398
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DNB|139092226
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NII|DA10092005
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BNF|11912066
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LC|nb2015007301
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996
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PLWABN|9810539782005606
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DNB|14322316X
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BIBSYS|2065405
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ISNI|0000000051924394
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ISNI|0000000505716566
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J9U|987007337315305171
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NTA|069361967
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NII|DA05393137
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ISNI|0000000430976645
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BIBSYS|4041696
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CAOONL|ncf12026805
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BIBSYS|90830379
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ISNI|0000000497275587
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NDL|00537740
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LC|n 92031795
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RERO|A006291501
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SUDOC|026978202
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ISNI|0000000504818173
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ISNI|0000000030085720
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LC|n 91116061
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J9U|987007343469305171
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LC|n 81030541
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|
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SUDOC|140465502
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996
|
|
|
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SUDOC|244875340
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996
|
|
|
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CAOONL|ncf11220625
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996
|
|
|
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BNF|15062094
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CAOONL|ncf10087942
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996
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NKC|jx20090720004
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996
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ISNI|0000000051483074
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NLA|000035297360
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NUKAT|n 01092785
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996
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ISNI|0000000063926741
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DNB|1124081720
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SUDOC|029275261
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996
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NUKAT|n 2021125824
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LC|no2024105193
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996
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NTA|070653054
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ISNI|0000000011171033
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ISNI|0000000045274954
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LC|n 86109924
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LC|n 2003104878
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ISNI|0000000512662359
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ISNI|0000000084434244
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CAOONL|ncf10125743
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J9U|987007588124205171
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RERO|A023803035
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ISNI|0000000374307294
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CAOONL|ncf11880858
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996
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ISNI|0000000122118075
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996
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PLWABN|9810640820405606
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LC|n 99050564
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ISNI|000000049300531X
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996
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CAOONL|ncf10348263
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996
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RERO|A009146821
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996
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ISNI|0000000495642128
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B2Q|0001261625
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ISNI|0000000455321311
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996
|
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LIH|LNB:CY_n__p_;=CK
|
996
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ISNI|0000000478942532
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996
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ISNI|0000000473564202
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ISNI|0000000108579676
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EGAXA|vtls001131099
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NII|DA13982756
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ISNI|0000000021710635
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NII|DA01211293
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LC|n 87926123
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DBC|87097969571743
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996
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LC|nb2018011315
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CAOONL|ncf10293525
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LC|nr 92035383
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ISNI|0000000114808324
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ISNI|0000000367927647
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BIBSYS|90565378
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LC|n 2021008736
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LC|n 79050920
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DNB|172220629
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ISNI|0000000483575570
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LC|n 85085616
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BIBSYS|97025375
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ISNI|0000000509839504
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LC|n 2020027712
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BNF|13936579
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UAE|Mill_a10001750
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SUDOC|129507970
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LC|n 81101449
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RERO|A014273031
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LC|no2015083636
|
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NLA|000035297350
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LC|n 2002063398
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JPG|500029906
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NKC|xx0227093
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LC|no 96006004
|
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|
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LC|n 82226796
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ISNI|0000000480120255
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BIBSYS|90345169
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NTA|06828795X
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ISNI|0000000033520564
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ISNI|0000000513671222
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NII|DA05537452
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RERO|A022809736
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ISNI|0000000367008210
|
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|
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NII|DA00763680
|
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|
|
|
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ISNI|0000000493194763
|
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|
|
|
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CYT|AC000006604
|
997
|
|
|
‡a
1900 0 flourished 0000 0
‡9
1
|